Tilfrinib

Tilfrinib

CAT N°: 25647
Price:

From 68.00 57.80

Tilfrinib is an inhibitor of breast tumor kinase/protein tyrosine kinase 6 (BRK/PTK6; IC50 = 3.15 nM).{42337,42338} It is selective for BRK/PTK6 over HER2 (IC50 = 1,300 nM).{42338} Tilfrinib inhibits the growth of MCF-7, HS-578/T, and BT-549 breast cancer cells in vitro (GI50s = 0.99, 1.02, and 1.58 ?M, respectively).{42337}

Territorial Availability: Available through Bertin Technologies only in France

  • Synonyms
    • 3-(9H-pyrido[2,3-b]indol-4-ylamino)-phenol
  • Correlated keywords
    • PTK-6 HER-2 MCF7 HS578 BT549 HS-578T HS578T
  • Product Overview:
    Tilfrinib is an inhibitor of breast tumor kinase/protein tyrosine kinase 6 (BRK/PTK6; IC50 = 3.15 nM).{42337,42338} It is selective for BRK/PTK6 over HER2 (IC50 = 1,300 nM).{42338} Tilfrinib inhibits the growth of MCF-7, HS-578/T, and BT-549 breast cancer cells in vitro (GI50s = 0.99, 1.02, and 1.58 ?M, respectively).{42337}

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