PSB-KD107

PSB-KD107

CAT N°: 31393
Price:

From 122.00 103.70

PSB-KD107 is an agonist of the orphan G protein-coupled receptor GPR18 (EC50 = 0.56 µM in a ?-arrestin recruitment assay using CHO cells expressing the human receptor).{58090,44024} It is selective for GPR18 over GPR55, as well as cannabinoid 1 (CB1) and CB2 receptors, at 10 µM but also binds to the adenosine A2A receptor (Ki = 0.33 µM for the rat receptor).{58090,58091}

Territorial Availability: Available through Bertin Technologies only in France

  • Synonyms
    • 6,7,8,9-tetrahydro-9-[2-(1H-indol-3-yl)ethyl]-1,3-dimethyl-pyrimido[2,1-f]purine-2,4(1H,3H)-dione
  • Correlated keywords
    • PSBKD107 GPR 18 55 CB 1 2 A 2A
  • Product Overview:
    PSB-KD107 is an agonist of the orphan G protein-coupled receptor GPR18 (EC50 = 0.56 µM in a ?-arrestin recruitment assay using CHO cells expressing the human receptor).{58090,44024} It is selective for GPR18 over GPR55, as well as cannabinoid 1 (CB1) and CB2 receptors, at 10 µM but also binds to the adenosine A2A receptor (Ki = 0.33 µM for the rat receptor).{58090,58091}

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