Propiverine (hydrochloride)

Propiverine (hydrochloride)

CAT N°: 36049
Price:

From 60.00 51.00

Propiverine is an antagonist of muscarinic acetylcholine receptors (mAChRs).{65340} It binds to M1 and M2 mAChRs in rat bladder and submaxillary gland, respectively (Kis = 0.3 and 0.19 µM, respectively), and inhibits carbachol-induced contraction of bladder strips isolated from patients with normal bladder activity and detrusor overactivity associated with benign prostatic hyperplasia (pA2s = 7.7 and 7.6, respectively).{65341} Formulations containing propiverine have been used in the treatment of overactive bladder.

Territorial Availability: Available through Bertin Technologies only in France

  • Synonyms
    • ?-phenyl-?-propoxy-benzeneacetic acid, 1-methyl-4-piperidinyl ester, monohydrochloride
  • Correlated keywords
    • 60569-19-9 anticholinergic anti-cholinergic Mictonetten Mictonorm P-4 P4 Pollarine mAChR pA2
  • Product Overview:
    Propiverine is an antagonist of muscarinic acetylcholine receptors (mAChRs).{65340} It binds to M1 and M2 mAChRs in rat bladder and submaxillary gland, respectively (Kis = 0.3 and 0.19 µM, respectively), and inhibits carbachol-induced contraction of bladder strips isolated from patients with normal bladder activity and detrusor overactivity associated with benign prostatic hyperplasia (pA2s = 7.7 and 7.6, respectively).{65341} Formulations containing propiverine have been used in the treatment of overactive bladder.

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