Volinanserin

Volinanserin

CAT N°: 15936
Price:

From 82.00 69.70

Volinanserin is a potent and selective antagonist of the serotonin receptor 5-HT2A (Ki = 0.36-0.85 nM).{25877,25875} It weakly binds 5-HT2C, ?1-adrenergic, and sigma receptors (Ki = 88, 128, and 87 nM) and much less effectively associates with other serotonin, dopamine, adrenergic, muscarinic acetylcholine receptors and monoamine transporters.{25875,25876} Volinanserin displays antipsychotic activity, attenuates impulsivity, and augments antidepressant effects in vivo.{25877,25878,23022}

Territorial Availability: Available through Bertin Technologies only in France

  • Synonyms
    • ?R-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-piperidinemethanol
  • Correlated keywords
    • receptors antagonists neurosciences selective serotonin 5-HT2A HT2A 5-HTs HTs 5 five 5HT2A potent MDLs 100907 MDL100907 MDL-100907 R-MDL RMDL R M antipsychotic impulsivity impulsive antidepressant (+)-MDL
  • Product Overview:
    Volinanserin is a potent and selective antagonist of the serotonin receptor 5-HT2A (Ki = 0.36-0.85 nM).{25877,25875} It weakly binds 5-HT2C, ?1-adrenergic, and sigma receptors (Ki = 88, 128, and 87 nM) and much less effectively associates with other serotonin, dopamine, adrenergic, muscarinic acetylcholine receptors and monoamine transporters.{25875,25876} Volinanserin displays antipsychotic activity, attenuates impulsivity, and augments antidepressant effects in vivo.{25877,25878,23022}

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