MRS1523

MRS1523

CAT N°: 17128
Price:

From 83.00 70.55

MRS1523 is an adenosine A3 receptor antagonist.{27929} It binds to the human adenosine A3 receptor (Ki = 0.0189 µM), as well as selectively binds rat adenosine A3 over A1 and A2A receptors (Kis = 0.113, 15.6, and 2.05 µM, respectively) in radioligand binding assays. It inhibits the proliferation of B16-BL6 mouse melanoma cells when used at a concentration of 1 µM.{68186}

Territorial Availability: Available through Bertin Technologies only in France

  • Synonyms
    • 6-ethyl-5-[(ethylthio)carbonyl]-2-phenyl-4-propyl-3-pyridinecarboxylic acid propyl ester
  • Correlated keywords
    • MRS 1523 radio ligand B16BL6
  • Product Overview:
    MRS1523 is an adenosine A3 receptor antagonist.{27929} It binds to the human adenosine A3 receptor (Ki = 0.0189 µM), as well as selectively binds rat adenosine A3 over A1 and A2A receptors (Kis = 0.113, 15.6, and 2.05 µM, respectively) in radioligand binding assays. It inhibits the proliferation of B16-BL6 mouse melanoma cells when used at a concentration of 1 µM.{68186}

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