24(S),25-epoxy Cholesterol
24(S),25-epoxy Cholesterol
24(S),25-epoxy Cholesterol is an oxysterol and the most abundant oxysterol in mouse ventral midbrain.{43943} It activates liver X receptors (LXRs)...
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From €102.00 €86.70
Melperone-d4 is intended for use as an internal standard for the quantification of melperone (Item No. 19770) by GC- or LC-MS. Melperone is an atypical antipsychotic.{25511} It binds to ?1- and ?2-adrenergic and dopamine D2 receptors (Kds = 180, 150, and 180 nM, respectively), as well as the serotonin (5-HT) receptor subtype 5-HT2A (Kd = 102 nM). It is selective for these receptors over histamine H1, muscarinic, 5-HT1A, 5-HT1D, and 5-HT2C receptors (Kds = 580, >10,000, 2,200, 3,400, and 2,100 nM, respectively). Melperone (2 mg/kg per day) increases basal, but not amphetamine-induced, extracellular dopamine levels in the rat nucleus accumbens.{53986}
Territorial Availability: Available through Bertin Technologies only in France
| Size | 1 mg, 5 mg, 500 µg |
|---|---|
| Shipping | dry ice |
| CAS number | 1219798-80-7 |
| Molecular formula | C16H18D4FNO • HCl |
| Smiles | CC(CC1([2H])[2H])CC([2H])([2H])N1CCCC(C2=CC=C(F)C=C2)=O.Cl |
| Molecular weight | 303,8 |
| Custom code | 3822.19 |
| Formulation | A solid |
| Purity | ≥99% deuterated forms (d1-d4) |
| UNSPSC code | 12352100 |
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