Adenosine Receptor A2A Blocking Peptide
Adenosine Receptor A2A Blocking Peptide
Adenosine Receptor A2A is a multi-pass membrane protein that is normally localized to the plasma membrane.{15465} This receptor is part...
€102.00 €86.70
Estradiol 3-(?-D-glucuronide) (E23G) is a non-cholestatic regioisomer of the estrogen metabolite, estradiol 17-(?-D-glucuronide) (E217G; Item No. 16156).{26342,26341} It acts as a substrate for multidrug resistance protein 2 (MRP2; Km = 122 µM), competing with E217G for MRP2-mediated transport (IC50 = 14.2 µM).{26341,26340} E23G has been reported to inhibit E217G transport through rat organic anion-transporting polypeptide 1 with a Ki value of 9.7 µM, but is a low-affinity inhibitor of both MRP4 and MRP7 (IC50s = ~ 100 µM).{26341}
Territorial Availability: Available through Bertin Technologies only in France
Size | 1 mg, 10 mg, 25 mg, 5 mg |
---|---|
Shipping | dry ice |
CAS number | 14982-12-8 |
Molecular formula | C24H31O8 • Na |
Smiles | [O-]C([C@H]([C@@H](O)[C@H](O)[C@H]1O)O[C@H]1OC2=CC=C3C(CC[C@]4([H])[C@]3([H])CC[C@@]5(C)[C@@]4([H])CC[C@@H]5O)=C2)=O.[Na+] |
Molecular weight | 470,5 |
Custom code | 2906.13 |
Formulation | A crystalline solid |
Purity | ≥95% |
UNSPSC code | 12352100 |
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Our scientists are experts in the synthesis, purification, and characterization of biochemicals ranging from small drug-like heterocycles to complex biolipids, fatty acids, and many others. We are also highly skilled in all aspects of assay and antibody development, protein expression, crystallization, and structure determination.
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Adenosine Receptor A2A is a multi-pass membrane protein that is normally localized to the plasma membrane.{15465} This receptor is part...
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