Enzastaurin

Enzastaurin

CAT N°: 11601
Price:

From 129.00 109.65

Enzastaurin is a potent inhibitor of PKC? (IC50 = 6 nM), with modest selectivity over PKC?, PKC?, and PKC? (IC50 = 39, 83, and 110 nM, respectively).{24308} At 3 µM, enzastaurin also inhibits signaling through the Akt pathway.{24306} It suppresses angiogenesis, induces apoptosis, and reduces proliferation of cultured tumor cells.{24308,24306} Because of these effects, enzastaurin has potential antineoplastic activity.{24307}

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