BMS 986188

BMS 986188

CAT N°: 21548
Price:

From 66.00 56.10

BMS 986188 is a positive allosteric modulator of ?-opioid receptors, with an EC50 value of 0.05 ?M in a ?-arrestin recruitment assay in the presence, but not absence, of the opioid receptor agonist leu-enkephalin (Item No. 23283).{38565} It is selective for ?- over ?-opioid receptors (EC50 = >10 ?M) in the presence of leu-enkephalin and the ?-opioid receptor agonist endomorphin 1 (Item No. 23280), respectively.

Territorial Availability: Available through Bertin Technologies only in France

  • Synonyms
    • 9-[4-[(2-bromophenyl)methoxy]phenyl]-3,4,5,6,7,9-hexahydro-3,3,6,6-tetramethyl-1H-xanthene-1,8(2H)-dione
  • Correlated keywords
    • BMS986188
  • Product Overview:
    BMS 986188 is a positive allosteric modulator of ?-opioid receptors, with an EC50 value of 0.05 ?M in a ?-arrestin recruitment assay in the presence, but not absence, of the opioid receptor agonist leu-enkephalin (Item No. 23283).{38565} It is selective for ?- over ?-opioid receptors (EC50 = >10 ?M) in the presence of leu-enkephalin and the ?-opioid receptor agonist endomorphin 1 (Item No. 23280), respectively.

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