Benzomalvin C

Benzomalvin C

CAT N°: 22064
Price:

779.00 662.15

Benzomalvin C is a weak antagonist of the neurokinin-1 (NK1) receptor inhibiting binding of substance P by 46% when used at 100 µg/ml in vitro.{38039} It is also a weak inhibitor of indolamine 2,3-dioxygenase (IDO) with an IC50 value of 130 µM for recombinant IDO.{38038} It was isolated from Penicillium and contains an epoxide group at C-19 and C-20, which is not present in benzomalvins A, B, or E.

Territorial Availability: Available through Bertin Technologies only in France

  • Synonyms
    • (2R,3S)-rel-(+)-6′-methyl-3-phenyl-spiro[oxirane-2,7′(13’H)-quinazolino[3,2-a][1,4]benzodiazepine]-5′,13′(6’H)-dione
  • Correlated keywords
    • NK-1 C19 C20
  • Product Overview:
    Benzomalvin C is a weak antagonist of the neurokinin-1 (NK1) receptor inhibiting binding of substance P by 46% when used at 100 µg/ml in vitro.{38039} It is also a weak inhibitor of indolamine 2,3-dioxygenase (IDO) with an IC50 value of 130 µM for recombinant IDO.{38038} It was isolated from Penicillium and contains an epoxide group at C-19 and C-20, which is not present in benzomalvins A, B, or E.

We also advise you