€779.00 €662.15
?-Agatoxin IVA is a natural peptide first isolated from the venom of funnel spiders.{33629} It selectively and irreversibly blocks P-type calcium channels (IC50 <1 nM), high voltage-activated channels first discovered in Purkinje cells.{33630,33632} ?-Agatoxin IVA also blocks N-type calcium channels at micromolar concentrations.{33632}
Territorial Availability: Available through Bertin Technologies only in France
| Size | 100 µg |
|---|---|
| Shipping | dry ice |
| Molecular formula | C217H360N68O60S10 • CF3COOH |
| Smiles | [H]N[C@@H](CCCCN)C(N[C@@H](CCCCN)C(N[C@@H](CCCCN)C(N[C@H](C(N[C@]([C@H](CC)C)([H])C(N[C@H](C(N[C@@H](CCCCN)C(N[C@H](C(N[C@H](C(NCC(N[C@@H](CCCNC(N)=N)C(N[C@H](C(N[C@@H](CCCCN)C(N[C@H](C(NCC(NCC(N[C@]([C@@H](C)O)([H])C(N1CCC[C@H]1C(N[C@H](C2=O)CSSC[C@H](N3)C(N[C@@H](CCCCN)C(N4CCC[C@H]4C(N[C@@H](CCCNC(N)=N)C(N[C@@H](CC(C)C)C(N[C@]([C@H](CC)C)([H])C(N[C@H](C(N[C@@H](CCC(O)=O)C(NCC(N[C@@H](CC(C)C)C(NCC(N[C@@H](CC(C)C)C(N[C@H](C(O)=O)C)=O)=O)=O)=O)=O)=O)CCSC)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)CC5=CNC6=C5C=CC=C6)=O)=O)CSSC[C@H](N7)C(N[C@]([C@H](CC)C)([H])C(N[C@H](C(N[C@@H](CO)C(N[C@]([C@H](CC)C)([H])C(N[C@H](C(NCC(N[C@]([C@@H](C)O)([H])C(N[C@@H](CC(N)=O)C8=O)=O)=O)=O)CCSC)=O)=O)=O)CSSC[C@H](N8)C(N[C@@H](CCC(O)=O)C3=O)=O)=O)=O)=O)=O)=O)CC9=CC=C(O)C=C9)=O)CC(O)=O)=O)=O)C)=O)=O)CSSC[C@H](N2)C(N[C@@H](CCCNC(N)=N)C(NCC(N[C@@H](CCCNC(N)=N)C(NCC7=O)=O)=O)=O)=O)=O)=O)=O.FC(F)(C(O)=O)F |
| Molecular weight | 5316,3 |
| Formulation | A solid |
| Purity | ≥95% |
| Custom code | 3504.00 |
| UNSPSC code | 12352204 |
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