CYM 2503

CYM 2503

CAT N°: 36590
Price:

From 66.00 56.10

CYM 2503 is a positive allosteric modulator (PAM) of the galanin-2 (GAL2) receptor.{64502} It enhances the production of inositol monophosphate (IP1) induced by galanin in HEK293 cells expressing the GAL2 receptor (EC50 = 0.69 µM). CYM 2503 (60 mg/kg) increases the latency to first electrographic and behavioral seizures and reduces mortality in a lithium-pilocarpine (Li-pilocarpine) rat model of status epilepticus.

Territorial Availability: Available through Bertin Technologies only in France

  • Synonyms
    • 3-cyclohexyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-alanyl-N-(1,2-dihydro-4-methyl-2-oxo-7-quinolinyl)-N6-[(1,1-dimethylethoxy)carbonyl]-L-lysinamide
  • Correlated keywords
    • CYM2503 HEK 293
  • Product Overview:
    CYM 2503 is a positive allosteric modulator (PAM) of the galanin-2 (GAL2) receptor.{64502} It enhances the production of inositol monophosphate (IP1) induced by galanin in HEK293 cells expressing the GAL2 receptor (EC50 = 0.69 µM). CYM 2503 (60 mg/kg) increases the latency to first electrographic and behavioral seizures and reduces mortality in a lithium-pilocarpine (Li-pilocarpine) rat model of status epilepticus.

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