CTAP (trifluoroacetate salt)

CTAP (trifluoroacetate salt)

CAT N°: 14959
Price:

213.00 181.05

CTAP is a water soluble, cyclic octapeptide which acts as a receptor antagonist that is selective for the µ opioid receptor (IC50 = 3.5 nM) over the ? receptor (IC50 = 4,500 nM).{23794} It is a poor antagonist of the somatostatin receptor (IC50 = 14.3 ?M).{23794} CTAP is at least 10-fold more potent than naltrexone as an antagonist of diverse compounds which have antinociceptive effects through the µ opioid receptor.{23793} It resists enzymatic metabolism in the blood and enters the brain and cerebrospinal fluid.{23791}

Territorial Availability: Available through Bertin Technologies only in France

  • Synonyms
    • D-phenylalanyl-L-cysteinyl-L-tyrosyl-D-tryptophyl-L-arginyl-L-threonyl-3-mercapto-L-valyl-cyclic (2?7)-disulfide-L-threoninamide, trifluoroacetate salt
  • Correlated keywords
    • 103429-32-9 cerebro-spinal octa-peptide TFA
  • Product Overview:
    CTAP is a water soluble, cyclic octapeptide which acts as a receptor antagonist that is selective for the µ opioid receptor (IC50 = 3.5 nM) over the ? receptor (IC50 = 4,500 nM).{23794} It is a poor antagonist of the somatostatin receptor (IC50 = 14.3 ?M).{23794} CTAP is at least 10-fold more potent than naltrexone as an antagonist of diverse compounds which have antinociceptive effects through the µ opioid receptor.{23793} It resists enzymatic metabolism in the blood and enters the brain and cerebrospinal fluid.{23791}

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