Nemonapride

Nemonapride

CAT N°: 21376
Price:

From 66.00 56.10

Nemonapride is an antipsychotic that readily passes through the blood brain barrier and exhibits potent neuroleptic effects in animals.{34046} It binds dopamine 2 (D2)-like receptors preferentially over D1-like receptors (Kis = 0.06, 0.3, and 0.15 nM for D2, D3, and D4, respectively).{34046,32473} Nemonapride also binds sigma 1 (?1) and ?2 receptors (Kis = 8.4 and 9.6 nM, respectively) and activates the serotonin 1A receptor (5-HT1A; IC50 = 34 nM).{34047,34045}

Territorial Availability: Available through Bertin Technologies only in France

  • Synonyms
    • rel-5-chloro-2-methoxy-4-(methylamino)-N-[(2R,3R)-2-methyl-1-(phenylmethyl)-3-pyrrolidinyl]-benzamide
  • Correlated keywords
    • 93664-94-9 emilace emonapride YM09151 YM09151-2 YM-09151 YM-091512 YM091512 anti-psychotic D2DR
  • Product Overview:
    Nemonapride is an antipsychotic that readily passes through the blood brain barrier and exhibits potent neuroleptic effects in animals.{34046} It binds dopamine 2 (D2)-like receptors preferentially over D1-like receptors (Kis = 0.06, 0.3, and 0.15 nM for D2, D3, and D4, respectively).{34046,32473} Nemonapride also binds sigma 1 (?1) and ?2 receptors (Kis = 8.4 and 9.6 nM, respectively) and activates the serotonin 1A receptor (5-HT1A; IC50 = 34 nM).{34047,34045}

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