2-<wbr/>furoyl-<wbr/>LIGRLO amide (trifluoroacetate salt)

2-furoyl-LIGRLO amide (trifluoroacetate salt)

CAT N°: 14594
Price:

174.00 147.90

2-furoyl-LIGRLO amide is a potent and selective agonist of the proteinase-activated receptor, PAR2 (pD2 = 7.0).{23092} It does not activate PAR1 or PAR4. Through its effects on PAR2, 2-furoyl-LIGRLO amide produces a concentration-dependent relaxation of arteries previously contracted with ?1 adrenergic receptor agonists.{23092}

Territorial Availability: Available through Bertin Technologies only in France

  • Synonyms
    • N-(2-furanylcarbonyl)-L-leucyl-L-isoleucylglycyl-L-arginyl-L-leucyl-L-ornithinamide, trifluoroacetate
  • Correlated keywords
    • 2468029-34-5 729589-58-6 receptors agonists vascular diseases inflammation potent PAR2 PAR-2 PARs 2 two amides LIGRLO furoyl selectives proteinase-activated proteinase activated active arteries a1 adrenergic a-1 a 1 alpha1 alpha-1 alpha .alpha.1 .alpha.-1 .alpha. ?1 ?-1 ? relaxation relax TFA
  • Product Overview:
    2-furoyl-LIGRLO amide is a potent and selective agonist of the proteinase-activated receptor, PAR2 (pD2 = 7.0).{23092} It does not activate PAR1 or PAR4. Through its effects on PAR2, 2-furoyl-LIGRLO amide produces a concentration-dependent relaxation of arteries previously contracted with ?1 adrenergic receptor agonists.{23092}

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